Therapeutic Forum

Be Heart-Smart 
When Treating the Eye

Christopher J. Quinn, O.D.

Read about "Coronary Heart Disease in the United States"

What’s your first choice of therapy for treating primary open angle glaucoma? If you’re thinking beta-blockers, you’re in good company. Today’s standard-of-practice for optometrists is to use a non-selective beta-blocker as the first line agent in the treatment of POAG.

This approach made perfect sense 15 years ago when we had only three topical agents to treat glaucoma. The two other agents were pilocarpine and epinephrine. Because of pilocarpine’s side effects and epinephrine’s high rate of allergic reactions, beta-blockers were the obvious choice.

But today we have more choices. These choices give us the opportunity and the responsibility to be more selective before prescribing a lifelong term of therapy. One consideration that merits your attention is the effect that beta-blockers—even topically applied—have on blood lipid levels.

True, studies and experience have shown that non-selective beta-blockers are dependable and effective in decreasing intraocular pressure. Side effects are well recognized, and careful patient selection can avoid most problems.

However, recent research has focused attention on beta-blockers’ ability to alter a patient’s serum lipid profile. Specifically, topical application of non-selective beta-blockers has been shown to reduce high-density lipoprotein (HDL) cholesterol levels (the “good” cholesterol component) and increase serum triglycerides. Decreased HDL and increased triglycerides can increase the risk of coronary heart disease and atherosclerosis. It’s thought that beta-blockers may alter blood lipid levels by inhibiting the enzyme lipoprotein lipase.

Ten years ago, researchers first described the effect of topical timolol 0.5% on patients with glaucoma and ocular hypertension.1 They found a statistically significant decrease in serum HDL and an increase in serum triglycerides. These authors predicted this change in blood lipids increased the risk of coronary artery disease by 21%.

The results have been confirmed in subsequent studies. Most recently, a comparative study of the effect of non-selective beta-blockers on blood lipid levels showed no significant difference between timolol maleate (Timoptic), carteolol hydrochloride (Ocupress) and metipranolol (Optipranolol) in their effect on blood lipid levels.2 This is significant since previous studies had indicated a potential benefit in the use of carteolol in its effect on blood lipid levels.

These studies prove one important thing: We need to consider the effect of our treatment on the patient’s general health as well as the local effect in reducing IOP. Long-term therapy, particularly in patients who have elevated cholesterol or other significant risk factors for coronary artery disease, may work better with an alternative agent as the initial treatment of choice.

Today’s alternatives—including alpha-agonists, prostaglandin analogs and carbonic anhydrase inhibitors—all can be effective in reducing IOP while not interfering with patients’ serum lipid levels.
 

1.Coleman et al. Topical timolol decreases plasma high-density lipoprotein cholesterol levels. Arch Ophthalmol 1990 Sep;108(9):1260-3.
2. Mirza GE et al. Comparison of the effects of 0.5% timolol maleate, 2% carteolol hydrochloride, and 0.3% metipranolol on intraocular pressure and perimetry findings and evaluation of their ocular and systemic effects. J Glaucoma 2000 Feb;9(1):45-50.

Coronary Heart Disease in the United States

  • CHD is the leading killer of American men and women.
  • 12 million Americans have a history of heart attack and/or angina.
  • Each year 1.1 million have heart attacks—370,000 die—250,000 die within 1 hour.
  • By age 60, every fifth man and 17th woman develops CHD (1986 Framingham data).
  • 1999 estimated direct and indirect costs of heart disease are $99.8 billion.
    —American Heart Association

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© Review of Optometry OnLine
April 15, 2000